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4-oxo-2-phenylmethanesulfonyl-octahydro-pyrrolo[1,2-a]pyrazine-6-carboxylic acid [1-(n-hydroxycarbamimidoyl)-piperidin-4-ylmethyl]-amide

Development stage
Unknown
Lead developer
Biochem Pharmaceutical Industries
Modality
Small Molecules
01

Overview

This compound is a synthetic small molecule dipeptide derivative with the molecular formula C22H32N6O5S and a molecular weight of approximately 492.6 g/mol. It is not approved for clinical use and is classified as an experimental agent in chemical databases. The structure features a pyrrolopyrazine core with sulfonamide and amidino substituents. According to available biochemical data, it acts as an inhibitor of thrombin (prothrombin), suggesting potential anticoagulant or antithrombotic activity; however, there are no known clinical indications or trials for this compound in humans[3][5][6].

Other names
(6S,8aS)-N-((1-((E)-N'-hydroxycarbamimidoyl)piperidin-4-yl)methyl)-4-oxo-2-phenylmethanesulfonyl-octahydropyrrolo(1,2-a)piperazine-6-carboxamide(6S,8aS)-N-{1-[E-N'-hydroxycarbamimidoyl]piperidin-4-yl}methyl)-4-oxo-2-phenyImethanesulfonyl-octahydropyrrolo[1,2-a]piperazine–6-carboxamide
02

Targets

F2 (Thrombin)

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